This book illustrates the influence of biomimetics in the field of tissue engineering and drug delivery. These two distinct fields of regenerative medicine have greatly benefited from the concept of biomimetics, which focuses on using or imitating nature to develop materials for improving human lives. The book begins by highlighting the relevance and recent advances in biomimetic biomaterials. An updated and innovative content has been presented in terms of biomimetic systems that are being utilized in controlled delivery and stem cell therapy. Further, the book reviews the role of these materials in enhanced capacity for drug loading, cellular uptake, and controlled release within the target cells. The book includes advanced techniques for characterizing biomimetic biomaterials and highlights their pivotal role in providing three-dimensional templates and synthetic extracellular matrices.